Phosphocreatine immobilization of the surface of silica and magnetite nanoparticles for targeted drug delivery


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A method is proposed for immobilization of anti-ischemic drug phosphocreatine on the surface of aminated silica and magnetite nanoparticles of similar size and shape. The synthesis of spacer and the coordination-ionic drug immobilization technique are described. Magnetite nanoparticles demonstrated much more efficient chemisorption of phosphocreatine than silica nanoparticles. The method was recommended for practical application.

作者简介

D. Korolev

Almazov National Medical Research Centre; First Pavlov State Medical University of St. Petersburg

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Email: Korolev_DV@almazovcentre.ru
俄罗斯联邦, 2 ul. Akkuratova, St. Petersburg, 197341; 6—8 ul. L’va Tolstogo, St. Petersburg, 197022

N. Evreinova

Almazov National Medical Research Centre; St. Petersburg State Technological Institute (Technical University)

Email: Korolev_DV@almazovcentre.ru
俄罗斯联邦, 2 ul. Akkuratova, St. Petersburg, 197341; 26 Moskovsky prosp., St. Petersburg, 190013

E. Zakharova

St. Petersburg Electrotechnical University “LETI”

Email: Korolev_DV@almazovcentre.ru
俄罗斯联邦, 5 ul. Prof. Popova, St. Petersburg, 197376

K. Gareev

St. Petersburg Electrotechnical University “LETI”

Email: Korolev_DV@almazovcentre.ru
俄罗斯联邦, 5 ul. Prof. Popova, St. Petersburg, 197376

E. Naumysheva

Almazov National Medical Research Centre; St. Petersburg State University

Email: Korolev_DV@almazovcentre.ru
俄罗斯联邦, 2 ul. Akkuratova, St. Petersburg, 197341; 7/9 Universitetskaya nab., St. Petersburg, 199034

D. Postnov

St. Petersburg State University

Email: Korolev_DV@almazovcentre.ru
俄罗斯联邦, 7/9 Universitetskaya nab., St. Petersburg, 199034

V. Postnov

Almazov National Medical Research Centre; St. Petersburg State University

Email: Korolev_DV@almazovcentre.ru
俄罗斯联邦, 2 ul. Akkuratova, St. Petersburg, 197341; 7/9 Universitetskaya nab., St. Petersburg, 199034

M. Galagudza

Almazov National Medical Research Centre; First Pavlov State Medical University of St. Petersburg

Email: Korolev_DV@almazovcentre.ru
俄罗斯联邦, 2 ul. Akkuratova, St. Petersburg, 197341; 6—8 ul. L’va Tolstogo, St. Petersburg, 197022

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