Modification of Automatic Synthesis of [18F]Fluoromisonidazole on a GE TracerLAB Fx F-N Synthesis Module


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Аннотация

A procedure for preparing 1-(2-hydroxy-3-[18F]fluoropropyl)-2-nitroimidazole ([18F]fluoromisonidazole, [18F]FMISO) on a commercially available GE TracerLAB Fx F-N synthesis module was developed. The product obtained meets all the requirements of the European Pharmacopoeia (8th ed.) for clinical use. Its decay-corrected radiochemical yield is 59 ± 4% (n = 5).

Авторлар туралы

D. Antuganov

Almazov Northwest Federal Medical Research Center

Хат алмасуға жауапты Автор.
Email: antuganov_do@almazovcentre.ru
Ресей, ul. Akkuratova 2, St. Petersburg, 197341

D. Ryzhkova

Almazov Northwest Federal Medical Research Center

Email: antuganov_do@almazovcentre.ru
Ресей, ul. Akkuratova 2, St. Petersburg, 197341

T. Zykova

Almazov Northwest Federal Medical Research Center

Email: antuganov_do@almazovcentre.ru
Ресей, ul. Akkuratova 2, St. Petersburg, 197341

V. Timofeev

Almazov Northwest Federal Medical Research Center

Email: antuganov_do@almazovcentre.ru
Ресей, ul. Akkuratova 2, St. Petersburg, 197341

Yu. Antuganova

Almazov Northwest Federal Medical Research Center

Email: antuganov_do@almazovcentre.ru
Ресей, ul. Akkuratova 2, St. Petersburg, 197341

K. Timofeeva

Almazov Northwest Federal Medical Research Center

Email: antuganov_do@almazovcentre.ru
Ресей, ul. Akkuratova 2, St. Petersburg, 197341

O. Samburov

Almazov Northwest Federal Medical Research Center

Email: antuganov_do@almazovcentre.ru
Ресей, ul. Akkuratova 2, St. Petersburg, 197341

M. Zykov

Almazov Northwest Federal Medical Research Center

Email: antuganov_do@almazovcentre.ru
Ресей, ul. Akkuratova 2, St. Petersburg, 197341

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