Four-Step Synthesis of Abiraterone Acetate from Dehydroepiandrosterone

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详细

A four-step synthesis of abiraterone acetate in good yield was developed. The synthesis employed Suzuki cross-coupling in the key step and produced the target compound in 99.8% purity.

作者简介

A. Balaev

Pharm-Sintez Co.

Email: chem@folium.ru
俄罗斯联邦, 8 2nd Roshchinskii Proezd, Moscow, 115419

A. Gromyko

Pharm-Sintez Co.

Email: chem@folium.ru
俄罗斯联邦, 8 2nd Roshchinskii Proezd, Moscow, 115419

V. Fedorov

Pharm-Sintez Co.

Email: chem@folium.ru
俄罗斯联邦, 8 2nd Roshchinskii Proezd, Moscow, 115419

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