Four-Step Synthesis of Abiraterone Acetate from Dehydroepiandrosterone
- Авторлар: Balaev A.N.1, Gromyko A.V.1, Fedorov V.E.1
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Мекемелер:
- Pharm-Sintez Co.
- Шығарылым: Том 50, № 6 (2016)
- Беттер: 404-406
- Бөлім: Drug Synthesis Methods and Manufacturing Technology
- URL: https://ogarev-online.ru/0091-150X/article/view/244404
- DOI: https://doi.org/10.1007/s11094-016-1459-1
- ID: 244404
Дәйексөз келтіру
Аннотация
A four-step synthesis of abiraterone acetate in good yield was developed. The synthesis employed Suzuki cross-coupling in the key step and produced the target compound in 99.8% purity.
Негізгі сөздер
Авторлар туралы
A. Balaev
Pharm-Sintez Co.
Email: chem@folium.ru
Ресей, 8 2nd Roshchinskii Proezd, Moscow, 115419
A. Gromyko
Pharm-Sintez Co.
Email: chem@folium.ru
Ресей, 8 2nd Roshchinskii Proezd, Moscow, 115419
V. Fedorov
Pharm-Sintez Co.
Email: chem@folium.ru
Ресей, 8 2nd Roshchinskii Proezd, Moscow, 115419
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