Hydroxamic acids: synthesis and adjuvant activity in combinatorial anticancer therapy


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Аннотация

Monoand disubstituted N-hydroxyamides of dicarboxylic acids were prepared by reaction of dicarboxylic acids or acid anhydrides with hydroxylamine. The use of these compounds in combinatorial cytostatic therapy of implanted tumors with cisplatin or cyclophosphamide totally inhibits metastasis formation in B16 melanoma and Lewis lung carcinoma, and resulted in 100% survival of leukemic animals.

Авторлар туралы

B. Fedorov

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Хат алмасуға жауапты Автор.
Email: boris-45@inbox.ru
Ресей, 1 prosp. Akad. N. N. Semenova, Chernogolovka, Moscow Region, 142432

M. Fadeev

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: boris-45@inbox.ru
Ресей, 1 prosp. Akad. N. N. Semenova, Chernogolovka, Moscow Region, 142432

A. Eremeev

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: boris-45@inbox.ru
Ресей, 1 prosp. Akad. N. N. Semenova, Chernogolovka, Moscow Region, 142432

N. Konovalova

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: boris-45@inbox.ru
Ресей, 1 prosp. Akad. N. N. Semenova, Chernogolovka, Moscow Region, 142432

G. Bogdanov

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: boris-45@inbox.ru
Ресей, 1 prosp. Akad. N. N. Semenova, Chernogolovka, Moscow Region, 142432

L. Tatyanenko

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: boris-45@inbox.ru
Ресей, 1 prosp. Akad. N. N. Semenova, Chernogolovka, Moscow Region, 142432

T. Sashenkova

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: boris-45@inbox.ru
Ресей, 1 prosp. Akad. N. N. Semenova, Chernogolovka, Moscow Region, 142432

D. Mishchenko

Institute of Problems of Chemical Physics, Russian Academy of Sciences

Email: boris-45@inbox.ru
Ресей, 1 prosp. Akad. N. N. Semenova, Chernogolovka, Moscow Region, 142432

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