Improved Process for Zoledronic Acid Synthesis


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Zoledronic acid is the drug substance of the highly efficient antiresorptive medicine Zometa. An improved synthesis of zoledronic acid via bis-phosphonation of 2-(1H-imidazol-1-yl)acetic acid is reported.

作者简介

Z. Kuvaeva

Institute of Physical Organic Chemistry, National Academy of Sciences of Belarus

Email: aminoacid1@ifoch.bas-net.by
白俄罗斯, Minsk

D. Lopatik

Institute of Physical Organic Chemistry, National Academy of Sciences of Belarus

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Email: aminoacid1@ifoch.bas-net.by
白俄罗斯, Minsk

O. Bondareva

Institute of Physical Organic Chemistry, National Academy of Sciences of Belarus

Email: aminoacid1@ifoch.bas-net.by
白俄罗斯, Minsk

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